N-Desmethylnefopam D5 hydrochloride

上海金畔生物科技有限公司为生命科学和医药研发人员提供生物活性分子抑制剂、激动剂、特异性抑制剂、化合物库、重组蛋白、同位素标记物,专注于信号通路和疾病研究领域。
N-Desmethylnefopam D5 hydrochloride 

N-Desmethylnefopam D5 hydrochloride 是 N-Desmethylnefopam hydrochloride 氘代物。N-Desmethylnefopam hydrochloride 是 Nefopam 的主要代谢产物,是一种中枢性但非阿片类化合物,可缓解中度至重度疼痛。

N-Desmethylnefopam D5 hydrochloride

N-Desmethylnefopam D5 hydrochloride Chemical Structure

规格 价格 是否有货
1 mg ¥2500 询问价格 & 货期
5 mg ¥5500 询问价格 & 货期

* Please select Quantity before adding items.

生物活性

N-Desmethylnefopam D5 hydrochloride is a deuterium labeled N-Desmethylnefopam hydrochloride. N-Desmethylnefopam hydrochloride is the main metabolite of Nefopam. N-Desmethylnefopam hydrochloride is a centrally-acting but non-opioid analgesic agent, for the relief of moderate to severe pain[1].

分子量

280.80

Formula

C16H13D5ClNO

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.

参考文献
  • [1]. Mittur A. A Simultaneous Mixed-Effects Pharmacokinetic Model for Nefopam, N-desmethylnefopam, and Nefopam N-Oxide in Human Plasma and Urine. Eur J Drug Metab Pharmacokinet. 2018 Aug;43(4):391-404.

所有产品仅用作科学研究或药证申报,我们不为任何个人用途提供产品和服务