3-Hydroxy agomelatine D3

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3-Hydroxy agomelatine D3 

3-Hydroxy agomelatine D3 是 3-Hydroxy agomelatine 的氘代物。3-Hydroxy agomelatine 是 5-HT2C 受体拮抗剂，IC50 为 3.2 μM，Ki 为 1.8 μM。

3-Hydroxy agomelatine D3

3-Hydroxy agomelatine D3 Chemical Structure

CAS No. : 1079774-23-4

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生物活性

3-Hydroxy agomelatine D3 is a deuterium labeled 3-Hydroxy agomelatine. 3-Hydroxy agomelatine is a 5-HT2C receptor antagonist with an IC50 of 3.2 μM and a Ki of 1.8 μM[1].

IC50 & Target[1]

5-HT2C Receptor

3.2 μM (IC50)

5-HT2C Receptor

1.8 μM (Ki)

分子量

262.32

Formula

C15H14D3NO3
CAS 号

1079774-23-4
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
参考文献

  • [1]. Chagraoui A, et al. Agomelatine(S 20098) antagonizes the penile erections induced by the stimulation of 5-HT2C receptors in Wistar rats. Psychopharmacology (Berl). 2003 Oct;170(1):17-22.

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