Mexiletine-d6 hydrochloride(Synonyms: KOE-1173-d6 hydrochloride)

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Mexiletine-d6 hydrochloride (Synonyms: KOE-1173-d6 hydrochloride) 纯度: ≥98.0%

Mexiletine D6 hydrochloride (KOE-1173 D6 hydrochloride) 是 Mexiletine hydrochloride (KOE-1173 hydrochloride) 的氘代物。Mexiletine hydrochloride,一种 Class IB 类抗心律失常化合物,是钠离子通道 (voltage-gated sodium channel) 阻断剂。

Mexiletine-d6 hydrochloride(Synonyms: KOE-1173-d6 hydrochloride)

Mexiletine-d6 hydrochloride Chemical Structure

CAS No. : 1329835-60-0

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10 mg ¥18000 In-stock
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生物活性

Mexiletine D6 hydrochloride (KOE-1173 D6 hydrochloride) is a deuterium labeled Mexiletine hydrochloride (KOE-1173 hydrochloride). Mexiletine hydrochloride, a Class IB antianhythmic, is a non-selective voltage-gated sodium channel blocker[1].

分子量

221.76

Formula

C11H12D6ClNO

CAS 号

1329835-60-0

中文名称

盐酸美西律 d6 (盐酸盐)

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

4°C, sealed storage, away from moisture

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

参考文献
  • [1]. Mori K, et al. Inhibitory effects of class I and IV antiarrhythmic drugs on the Na+-activated K+ channel current in guinea pig ventricular cells. Naunyn Schmiedebergs Arch Pharmacol. 1998 Dec;358(6):641-8.

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